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SAR125884 hydrochlorid
CAS No. ——
SAR125884 hydrochlorid ( —— )
Catalog No. M20372 CAS No. ——
SAR125844 is a potent and selective MET kinase inhibitor with a favorable preclinical toxicity profile(IC50=4.2 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 101 | Get Quote |
|
| 10MG | 168 | Get Quote |
|
| 25MG | 361 | Get Quote |
|
| 50MG | 687 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameSAR125884 hydrochlorid
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NoteResearch use only, not for human use.
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Brief DescriptionSAR125844 is a potent and selective MET kinase inhibitor with a favorable preclinical toxicity profile(IC50=4.2 nM).
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DescriptionSAR125844 is a potent and selective MET kinase inhibitor with a favorable preclinical toxicity profile(IC50=4.2 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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Targetc-Met/HGFR
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RecptorMET RTK
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight550.6
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Molecular FormulaC25H23FN8O2S2?
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.Fc1ccc(cc1)-c1ccc2nnc(Sc3ccc4nc(NC(=O)NCCN5CCOCC5)sc4c3)n2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.The Selective Intravenous Inhibitor of the MET Tyrosine Kinase SAR125844 Inhibits Tumor Growth in MET-Amplified Cancer[J]. Molecular Cancer Therapeutics 2015 14(2):384-394.
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